C29H27F2N7O5S
623.6 g/mol
APIDanger
Relugolix
CAS737789-87-6
Category
API
Compound Class
Heterocycle
Primary Use
Pharmaceutical Raw Material
Relugolix is a gonadotropin-releasing hormone (GnRH) receptor antagonist used as a pharmaceutical raw material. It is notable as the first orally administered GnRH receptor antagonist approved for advanced prostate cancer, offering a less burdensome option compared to injectable therapies.
Pharmaceutical manufacturing of GnRH receptor antagonist therapiesResearch compound for hormone-responsive conditionsActive pharmaceutical ingredient in combination products for uterine fibroids
Content scope: Information here supports chemical identification and industrial supply, research, and manufacturing contexts. It is not a therapeutic claim, medical advice, or drug-use instructions.
Sourcing Relugolix?
Post a free purchase request — no account needed. It reaches suppliers of this product, and replies go straight to your inbox.
Related Compounds
SimilarStructure SimilarSimilarity 0.80
6-(4-aminophenyl)-1-((2,6-difluorophenyl)methyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)thieno(2,3-d)pyrimidine-2,4(1H,3H)-dione
CAS1589503-93-4
pharmaceutical intermediate
SimilarStructure SimilarSimilarity 0.73
Thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione, 1-[(2,6-difluorophenyl)methyl]-5-[(dimethylamino)methyl]-3-(6-methoxy-3-pyridazinyl)-6-(4-nitrophenyl)-
CAS1589503-96-7
pharmaceutical intermediate
ReferenceSame Category
Trimethoprim
CAS738-70-5
pharmaceutical raw material
ReferenceSame Category
Trans-tramadol hydrochloride
CAS73806-49-2
pharmaceutical raw material
ReferenceSame Category
1,2-dehydro tramadol
CAS73825-64-6
pharmaceutical raw material
ReferenceSame Category
Trans-calcitriol
CAS73837-24-8
pharmaceutical raw material
Safety Reference
Danger
H360May damage fertility or the unborn child
H361Suspected of damaging fertility or the unborn child
H371May cause damage to organs
H373May cause damage to organs through prolonged or repeated exposure
H411Toxic to aquatic life with long lasting effects
Customs Tariff Classification
The international HS code for Relugolix (CAS 737789-87-6) is 2934.99.
HS code (international, 6-digit)
2934.99
EU CN code (8-digit)
2934 99 90
Classification per the EU customs inventory ECICS (2026-07 snapshot, HS 2022). National tariff lines and product form can affect the final classification.
Identifiers
IUPAC Name
1-[4-[1-[(2,6-difluorophenyl)methyl]-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-3-methoxyurea
InChIKey
AOMXMOCNKJTRQP-UHFFFAOYSA-N
SMILES
CN(C)CC1=C(SC2=C1C(=O)N(C(=O)N2CC3=C(C=CC=C3F)F)C4=NN=C(C=C4)OC)C5=CC=C(C=C5)NC(=O)NOC
Synonyms (20)
- TAK-385
- Relugolix (JAN/USAN/INN)
- MYFEMBREE COMPONENT RELUGOLIX
- Orgovyx
- Orgovyx (TN)
- Relugolix
- Relugolix (Standard)
- Relugolix(TAK-385)
- TAK-385; RVT-601
- relugolixum
Sourcing Relugolix?
Post a free purchase request — no account needed. It reaches suppliers of this product, and replies go straight to your inbox.