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Home/Compounds/Pharmaceutical Intermediate/N-(3-Chloro-4-fluorophenyl)-7-methoxy-6-nitroquinazolin-4-amine
C15H10ClFN4O3
348.71 g/mol
Pharmaceutical Intermediate

N-(3-Chloro-4-fluorophenyl)-7-methoxy-6-nitroquinazolin-4-amine

CAS179552-74-0
Category
Pharmaceutical Intermediate
Compound Class
Amine
Primary Use
Pharmaceutical Intermediate

N-(3-chloro-4-fluorophenyl)-7-methoxy-6-nitroquinazolin-4-amine is a quinazoline derivative used as a pharmaceutical intermediate. Its primary significance lies in its role as a building block in the synthesis of kinase inhibitors for research and manufacturing purposes.

Pharmaceutical intermediate for kinase inhibitor synthesis

Content scope: Information here supports chemical identification and industrial supply, research, and manufacturing contexts. It is not a therapeutic claim, medical advice, or drug-use instructions.

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SimilarStructure SimilarSimilarity 0.73

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Identifiers
IUPAC Name

N-(3-chloro-4-fluorophenyl)-7-methoxy-6-nitroquinazolin-4-amine

InChIKey

VKEKKVCWODTGAP-UHFFFAOYSA-N

SMILES

COC1=C(C=C2C(=C1)N=CN=C2NC3=CC(=C(C=C3)F)Cl)[N+](=O)[O-]

Synonyms (9)
  • Afatinib Impurity 5
  • Afatinib Impurity 89
  • Dacomitinib Intermediate 2