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Ana Sayfa/Bileşikler/Diğer/SuO-Glu-Val-Cit-PAB-MMAE
C67H103N11O17
1334.6 g/mol
Diğer

SuO-Glu-Val-Cit-PAB-MMAE

CAS1895916-24-1
Kategori
Diğer
Bileşik Sınıfı
Peptit
Birincil Kullanım
antibody-drug conjugate linker payload

This compound is an antibody-drug conjugate linker payload, composed of a cleavable linker and the antimitotic agent monomethyl auristatin E (MMAE). It is designed for use in the development of targeted cancer therapeutics.

research reagent for antibody-drug conjugate developmentcompound used in pharmaceutical manufacturing of targeted therapies

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Tanımlayıcılar
IUPAC Adı

(2,5-dioxopyrrolidin-1-yl) 5-[[(2S)-1-[[(2S)-5-(carbamoylamino)-1-[4-[[[(2S)-1-[[(2S)-1-[[(3R,4S,5S)-1-[(2S)-2-[(1R,2R)-3-[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]amino]-1-methoxy-2-methyl-3-oxopropyl]pyrrolidin-1-yl]-3-methoxy-5-methyl-1-oxoheptan-4-yl]-methylamino]-3-methyl-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-methylcarbamoyl]oxymethyl]anilino]-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-5-oxopentanoate

InChIKey

QULAXLHJSKOZMO-FBMBWUFNSA-N

SMILES

CC[C@H](C)[C@@H]([C@@H](CC(=O)N1CCC[C@H]1[C@@H]([C@@H](C)C(=O)N[C@H](C)[C@H](C2=CC=CC=C2)O)OC)OC)N(C)C(=O)[C@H](C(C)C)NC(=O)[C@H](C(C)C)N(C)C(=O)OCC3=CC=C(C=C3)NC(=O)[C@H](CCCNC(=O)N)NC(=O)[C@H](C(C)C)NC(=O)CCCC(=O)ON4C(=O)CCC4=O

Eş Anlamlılar (3)
  • OSU-VC-PAB-MMAE
  • OSu-Glu-vc-PAB-MMAE
  • SuO-Glu-Val-Cit-PAB-MMAE