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홈/화합물/원료의약품/B-[(1R)-3-Methyl-1-[[(2R)-1-oxo-3-phenyl-2-[(2-pyrazinylcarbonyl)amino]propyl]amino]butyl]boronic Acid
C19H25BN4O4
384.2 g/mol
원료의약품

B-[(1R)-3-Methyl-1-[[(2R)-1-oxo-3-phenyl-2-[(2-pyrazinylcarbonyl)amino]propyl]amino]butyl]boronic Acid

CAS1132709-15-9
용도 분류
원료의약품
화합물 분류
펩타이드
주요 용도
의약 원료

This compound is a boronic acid derivative featuring a pyrazine-2-carbonylamino group and a phenylalanine-like backbone. It is used as an active pharmaceutical ingredient in pharmaceutical manufacturing and research.

콘텐츠 범위: 이 페이지의 정보는 화학물질 식별 및 산업 공급·연구개발·제조 맥락을 대상으로 합니다. 치료 효능 주장, 의료 조언 또는 의약품 사용 지침에 해당하지 않습니다.

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보르테조밉

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참고same scaffold

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Pharmaceutical intermediate

참고same scaffold

N-(pyrazine-2-yl-carbonyl)-L-phenylalanine

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참고same scaffold

5-methyl-N-[2-(4-sulfamoylphenyl)ethyl]pyrazine-2-carboxamide

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식별자
IUPAC 이름

[(1R)-3-methyl-1-[[(2R)-3-phenyl-2-(pyrazine-2-carbonylamino)propanoyl]amino]butyl]boronic acid

InChIKey

GXJABQQUPOEUTA-WBVHZDCISA-N

SMILES

B([C@H](CC(C)C)NC(=O)[C@@H](CC1=CC=CC=C1)NC(=O)C2=NC=CN=C2)(O)O

동의어 목록 (12)
  • Boronic acid, B-[(1R)-3-methyl-1-[[(2R)-1-oxo-3-phenyl-2-[(2-pyrazinylcarbonyl)amino]propyl]amino]butyl]-; B-[(1R)-3-Methyl-1-[[(2R)-1-oxo-3-phenyl-2-[(2-pyrazinylcarbonyl)amino]propyl]amino]butyl]boronic acid; bortezomib diastereomer (R,R) (USP); bortezomib related compound A (USP)
  • (1R,2R)-Bortezomib
  • (1R,2R)-Bortezomib (>85%)
  • Bortezomib (1R, 2R)-Isomer
  • Bortezomib Impurity 7
  • Bortezomib, (1R,2R)-